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Activation loop targeting strategy for design of receptor-interacting protein kinase 2 (RIPK2) inhibitors

Development of selective kinase inhibitors remains a challenge due to considerable amino acid sequence similarity among family members particularly in the ATP binding site. Targeting the activation loop might offer improved inhibitor selectivity since this region of kinases is less conserved. Howeve...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Suebsuwong, Chalada, Pinkas, Daniel M., Ray, Soumya S., Bufton, Joshua C., Dai, Bing, Bullock, Alex N., Degterev, Alexei, Cuny, Gregory D.
Formato: Artigo
Idioma:Inglês
Publicado em: Elsevier Science Ltd 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5819902/
https://ncbi.nlm.nih.gov/pubmed/29409752
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.01.044
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