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Small molecule anionophores promote transmembrane anion permeation matching CFTR activity

Anion selective ionophores, anionophores, are small molecules capable of facilitating the transmembrane transport of anions. Inspired in the structure of natural product prodigiosin, four novel anionophores 1a-d, including a 1,2,3-triazole group, were prepared. These compounds proved highly efficien...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Hernando, Elsa, Capurro, Valeria, Cossu, Claudia, Fiore, Michele, García-Valverde, María, Soto-Cerrato, Vanessa, Pérez-Tomás, Ricardo, Moran, Oscar, Zegarra-Moran, Olga, Quesada, Roberto
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5805763/
https://ncbi.nlm.nih.gov/pubmed/29422673
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-20708-3
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