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Integrating Transcriptomic Data with Mechanistic Systems Pharmacology Models for Virtual Drug Combination Trials

Monotherapy clinical trials with mutation-targeted kinase inhibitors, despite some success in other cancers, have yet to impact glioblastoma (GBM). Besides insufficient blood-brain-barrier penetration, combinations are key to overcoming obstacles such as intratumoral heterogeneity, adaptive resistan...

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Detalles Bibliográficos
Publicado en:ACS Chem Neurosci
Autores principales: Barrette, Anne Marie, Bouhaddou, Mehdi, Birtwistle, Marc R.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5771884/
https://ncbi.nlm.nih.gov/pubmed/28950062
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00197
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