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Click Chemistry in Lead Optimization of Boronic Acids as β-Lactamase Inhibitors

Boronic acid transition state inhibitors (BATSIs) represent one of the most promising class of β-lactamase inhibitors. Here we describe a new class of BATSIs, namely 1-amido-2-triazolylethaneboronic acids, which were synthesized combining the asymmetric homologation of boronates with Copper-Catalyze...

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Détails bibliographiques
Publié dans:J Med Chem
Auteurs principaux: Caselli, Emilia, Romagnoli, Chiara, Vahabi, Roza, Taracila, Magdalena A., Bonomo, Robert A., Prati, Fabio
Format: Artigo
Langue:Inglês
Publié: 2015
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5744665/
https://ncbi.nlm.nih.gov/pubmed/26102369
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b00341
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