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Development of Phenyl Cyclohexylcarboxamides as a Novel Class of Hsp90 C-terminal Inhibitors

Inhibition of the heat shock protein 90 (Hsp90) C-terminus represents a promising therapeutic strategy for the treatment of cancer. Novobiocin, a coumarin antibiotic, was the first Hsp90 C-terminal inhibitor identified, however, it manifested poor anti-proliferative activity (SKBr3, IC(50) ~ 700 μM)...

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Detalhes bibliográficos
Publicado no:Chemistry
Main Authors: Garg, Gaurav, Forsberg, Leah K., Zhao, Huiping, Blagg, Brian S. J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5724527/
https://ncbi.nlm.nih.gov/pubmed/28940589
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.201703206
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