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Allosteric Tuning of Caspase‐7: A Fragment‐Based Drug Discovery Approach

The caspase family of cysteine proteases are highly sought‐after drug targets owing to their essential roles in apoptosis, proliferation, and inflammation pathways. High‐throughput screening efforts to discover inhibitors have gained little traction. Fragment‐based screening has emerged as a powerfu...

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Bibliographische Detailangaben
Veröffentlicht in:Angew Chem Int Ed Engl
Hauptverfasser: Vance, Nicholas R., Gakhar, Lokesh, Spies, M. Ashley
Format: Artigo
Sprache:Inglês
Veröffentlicht: John Wiley and Sons Inc. 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5698726/
https://ncbi.nlm.nih.gov/pubmed/28940929
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201706959
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