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A novel C-terminal HSP90 inhibitor KU135 induces apoptosis and cell cycle arrest in melanoma cells

Heat shock protein 90 (Hsp90) is differentially expressed in tumor cells including melanoma and involved in proper folding, stabilization and regulation of cellular proteins. We investigated a novobiocin-derived Hsp90 C-terminal inhibitor, KU135, for anti-proliferative effects in melanoma cells. The...

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Detalhes bibliográficos
Publicado no:Cancer Lett
Main Authors: Samadi, Abbas K., Zhang, Xuan, Mukerji, Ridhwi, Donnelly, Alison C., Blagg, Brian S., Cohen, Mark S.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5683962/
https://ncbi.nlm.nih.gov/pubmed/21924824
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.canlet.2011.07.031
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