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A novel C-terminal HSP90 inhibitor KU135 induces apoptosis and cell cycle arrest in melanoma cells

Heat shock protein 90 (Hsp90) is differentially expressed in tumor cells including melanoma and involved in proper folding, stabilization and regulation of cellular proteins. We investigated a novobiocin-derived Hsp90 C-terminal inhibitor, KU135, for anti-proliferative effects in melanoma cells. The...

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Publicat a:Cancer Lett
Autors principals: Samadi, Abbas K., Zhang, Xuan, Mukerji, Ridhwi, Donnelly, Alison C., Blagg, Brian S., Cohen, Mark S.
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5683962/
https://ncbi.nlm.nih.gov/pubmed/21924824
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.canlet.2011.07.031
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