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Evaluation of DILI Predictive Hypotheses in Early Drug Development

Drug-induced liver injury (DILI) is a leading cause of drug failure in clinical trials and a major reason for drug withdrawals. DILI has been shown to be dependent on both daily dose and extent of hepatic metabolism. Yet, early in drug development daily dose is unknown. Here, we perform a comprehens...

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Vydáno v:Chem Res Toxicol
Hlavní autoři: Chan, Rosa, Benet, Leslie Z.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2017
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5674994/
https://ncbi.nlm.nih.gov/pubmed/28257576
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.chemrestox.7b00025
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