Lanean...

Cytochrome b(5) plays a dual role in the reaction cycle of cytochrome P450 3A4 during oxidation of the anticancer drug ellipticine

ABSTRACT: Ellipticine is an anticancer agent that forms covalent DNA adducts after enzymatic activation by cytochrome P450 (CYP) enzymes, mainly by CYP3A4. This process is one of the most important ellipticine DNA-damaging mechanisms for its antitumor action. Here, we investigated the efficiencies o...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Monatsh Chem
Egile Nagusiak: Stiborová, Marie, Indra, Radek, Frei, Eva, Kopečková, Kateřina, Schmeiser, Heinz H., Eckschlager, Tomáš, Adam, Vojtěch, Heger, Zbyněk, Arlt, Volker M., Martínek, Václav
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Springer Vienna 2017
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC5653753/
https://ncbi.nlm.nih.gov/pubmed/29104319
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00706-017-1986-9
Etiketak: Etiketa erantsi
Etiketarik gabe, Izan zaitez lehena erregistro honi etiketa jartzen!