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Structural Determinants for the Selectivity of the Positive KCa3.1 Gating Modulator 5-Methylnaphtho[2,1-d]oxazol-2-amine (SKA-121)

Intermediate-conductance (K(Ca)3.1) and small-conductance (K(Ca)2) calcium-activated K(+) channels are gated by calcium binding to calmodulin (CaM) molecules associated with the calmodulin-binding domain (CaM-BD) of these channels. The existing K(Ca) activators, such as naphtho[1,2-d]thiazol-2-ylami...

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Shranjeno v:
Bibliografske podrobnosti
izdano v:Mol Pharmacol
Main Authors: Brown, Brandon M., Shim, Heesung, Zhang, Miao, Yarov-Yarovoy, Vladimir, Wulff, Heike
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5588545/
https://ncbi.nlm.nih.gov/pubmed/28760780
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.117.109421
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