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Structural Insights into the Atomistic Mechanisms of Action of Small Molecule Inhibitors Targeting the KCa3.1 Channel Pore

The intermediate-conductance Ca(2+)-activated K(+) channel (KCa3.1) constitutes an attractive pharmacological target for immunosuppression, fibroproliferative disorders, atherosclerosis, and stroke. However, there currently is no available crystal structure of this medically relevant channel that co...

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Détails bibliographiques
Publié dans:Mol Pharmacol
Auteurs principaux: Nguyen, Hai M., Singh, Vikrant, Pressly, Brandon, Jenkins, David Paul, Wulff, Heike, Yarov-Yarovoy, Vladimir
Format: Artigo
Langue:Inglês
Publié: The American Society for Pharmacology and Experimental Therapeutics 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5363711/
https://ncbi.nlm.nih.gov/pubmed/28126850
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.116.108068
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