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Targeted Protein Degradation by Small Molecules

Protein homeostasis networks are highly regulated systems responsible for maintaining the health and productivity of cells. Whereas therapeutics have been developed to disrupt protein homeostasis, more recently identified techniques have been used to repurpose homeostatic networks to effect degradat...

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Библиографические подробности
Опубликовано в: :Annu Rev Pharmacol Toxicol
Главные авторы: Bondeson, Daniel P., Crews, Craig M.
Формат: Artigo
Язык:Inglês
Опубликовано: 2016
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5586045/
https://ncbi.nlm.nih.gov/pubmed/27732798
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1146/annurev-pharmtox-010715-103507
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