Caricamento...

Effect of solvent and protein dynamics in ligand recognition and inhibition of aminoglycoside adenyltransferase 2″‐Ia

The aminoglycoside modifying enzyme (AME) ANT(2″)‐Ia is a significant target for next generation antibiotic development. Structural studies of a related aminoglycoside‐modifying enzyme, ANT(3″)(9), revealed this enzyme contains dynamic, disordered, and well‐defined segments that modulate thermodynam...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Protein Sci
Autori principali: Bacot‐Davis, Valjean R., Bassenden, Angelia V., Sprules, Tara, Berghuis, Albert M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2017
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5563142/
https://ncbi.nlm.nih.gov/pubmed/28734024
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/pro.3224
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !