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Autoinhibitory properties of the parent but not of the N‐oxide metabolite contribute to infusion rate‐dependent voriconazole pharmacokinetics

AIMS: The pharmacokinetics of voriconazole show a nonlinear dose–exposure relationship caused by inhibition of its own CYP3A‐dependent metabolism. Because the magnitude of autoinhibition also depends on voriconazole concentrations, infusion rate might modulate voriconazole exposure. The impact of fo...

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Detalles Bibliográficos
Publicado en:Br J Clin Pharmacol
Main Authors: Hohmann, Nicolas, Kreuter, Rebecca, Blank, Antje, Weiss, Johanna, Burhenne, Jürgen, Haefeli, Walter E., Mikus, Gerd
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5555860/
https://ncbi.nlm.nih.gov/pubmed/28370390
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcp.13297
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