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(125)I-4-Aminobenzyl-5′-N-methylcarboxamidoadenosine, a High Affinity Radioligand for the Rat A(3) Adenosine Receptor

The rat A(3) adenosine receptor (AR) is a recently characterized AR subtype cloned from testis and brain cDNA libraries. N(6)-2-(4-Amino-3-[(125)I]iodophenyl)ethyladenosine, a high affinity A(1)AR agonist, has served as the only radioligand available for study of the A(3)AR. The relatively low affin...

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Dettagli Bibliografici
Pubblicato in:Mol Pharmacol
Autori principali: OLAH, MARK E., GALLO-RODRIGUEZ, CAROLA, JACOBSON, KENNETH A., STILES, GARY L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1994
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5553074/
https://ncbi.nlm.nih.gov/pubmed/8190112
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