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A SELECTIVE AGONIST AFFINITY LABEL FOR A(3) ADENOSINE RECEPTORS

A newly synthesized, chemically reactive adenosine derivative, N(6)-(3-isothiocyanatobenzyl)adenosine-5'-N-methyluronamide, was found to bind selectively to A(3) receptors. K(i) values for this isothiocyanate derivative in competition binding at rat brain A(1), A(2a), and A(3) receptors were 14...

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Dettagli Bibliografici
Autori principali: Ji, Xiao-duo, Gallo-Rodriguez, Carola, Jacobson, Kenneth A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1994
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3425636/
https://ncbi.nlm.nih.gov/pubmed/8074705
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