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Structure-based identification of inhibitors targeting obstruction of the HIVgp41 N-Heptad repeat trimer

The viral protein HIVgp41 is an attractive and validated drug target that proceeds through a sequence of conformational changes crucial for membrane fusion, which facilitates viral entry. Prior work has identified inhibitors that interfere with the formation of a required six-helix bundle, composed...

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Shranjeno v:
Bibliografske podrobnosti
izdano v:Bioorg Med Chem Lett
Main Authors: McGee, T. Dwight, Yi, Hyun Ah, Allen, William J., Jacobs, Amy, Rizzo, Robert C.
Format: Artigo
Jezik:Inglês
Izdano: 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5551449/
https://ncbi.nlm.nih.gov/pubmed/28558972
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2017.05.020
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