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Potent Prearranged Positive Allosteric Modulators of the Glucagon‐like Peptide‐1 Receptor

Drugs that allosterically modulate G protein‐coupled receptor (GPCR) activity display higher specificity and may improve disease treatment. However, the rational design of compounds that target the allosteric site is difficult, as conformations required for receptor activation are poorly understood....

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Détails bibliographiques
Publié dans:ChemistryOpen
Auteurs principaux: Jones, Ben J., Scopelliti, Rosario, Tomas, Alejandra, Bloom, Stephen R., Hodson, David J., Broichhagen, Johannes
Format: Artigo
Langue:Inglês
Publié: John Wiley and Sons Inc. 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5542757/
https://ncbi.nlm.nih.gov/pubmed/28794944
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/open.201700062
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