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Synthetic analogues of migrastatin that inhibit mammary tumor metastasis in mice

Tumor metastasis is the most common cause of death in cancer patients. Here, we show that two, fully synthetic migrastatin analogues, core macroketone and core macrolactam, are potent inhibitors of metastasis in a murine breast tumor model. Administration of these readily accessible compounds nearly...

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Autors principals: Shan, Dandan, Chen, Lin, Njardarson, Jon T., Gaul, Christoph, Ma, Xiaojing, Danishefsky, Samuel J., Huang, Xin-Yun
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2005
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC553334/
https://ncbi.nlm.nih.gov/pubmed/15728385
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0500658102
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