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Somatic cancer mutations in the MLL1 histone methyltransferase modulate its enzymatic activity and dependence on the WDR5/RBBP5/ASH2L complex

Somatic missense mutations in the mixed lineage leukemia 1 (MLL1) histone H3K4 methyltransferase are often observed in cancers. MLL1 forms a complex with WDR5, RBBP5, and ASH2L (WRA) which stimulates its activity. The MM‐102 compound prevents the interaction between MLL1 and WDR5 and functions as an...

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Bibliografiset tiedot
Julkaisussa:Mol Oncol
Päätekijät: Weirich, Sara, Kudithipudi, Srikanth, Jeltsch, Albert
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: John Wiley and Sons Inc. 2017
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC5527479/
https://ncbi.nlm.nih.gov/pubmed/28182322
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/1878-0261.12041
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