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Valnoctamide, which reduces rat brain arachidonic acid turnover, is a potential non-teratogenic valproate substitute to treat bipolar disorder

BACKGROUND: Valproic acid (VPA), used for treating bipolar disorder (BD), is teratogenic by inhibiting histone deacetylase. In unanaesthetized rats, chronic VPA, like other mood stabilizers, reduces arachidonic acid (AA) turnover in brain phospholipids, and inhibits AA activation to AA-CoA by recomb...

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Dades bibliogràfiques
Publicat a:Psychiatry Res
Autors principals: Modi, Hiren R., Ma, Kaizong, Chang, Lisa, Chen, Mei, Rapoport, Stanley I.
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5524208/
https://ncbi.nlm.nih.gov/pubmed/28500975
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.psychres.2017.04.048
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