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Valnoctamide, a non-teratogenic amide derivative of valproic acid, inhibits arachidonic acid activation in vitro by recombinant acyl-CoA synthetase-4
OBJECTIVE: Valproic acid (VPA), a mood stabilizer used for treating bipolar disorder (BD), uncompetitively inhibits acylation of arachidonic acid (AA) by recombinant AA-selective acyl-CoA synthetase (Acsl)-4 at K(i) of 25 mM. Inhibition may account for VPA’s ability to reduce AA turnover in brain ph...
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| Publicado no: | Bipolar Disord |
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| Main Authors: | , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
2014
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4554599/ https://ncbi.nlm.nih.gov/pubmed/25041123 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bdi.12220 |
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