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Novel anti-inflammatory agents targeting CXCR4: Design, synthesis, biological evaluation and preliminary pharmacokinetic study

CXCR4 plays a crucial role in the inflammatory disease process, providing an attractive means for drug targeting. A series of novel amide-sulfamide derivatives were designed, synthesized and comprehensively evaluated. This new scaffold exhibited much more potent CXCR4 inhibitory activity, with more...

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Publicado en:Eur J Med Chem
Autores principales: Bai, Renren, Liang, Zhongxing, Yoon, Younghyoun, Salgado, Eric, Feng, Amber, Gurbani, Saumya, Shim, Hyunsuk
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5521218/
https://ncbi.nlm.nih.gov/pubmed/28521261
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2017.05.030
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