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The small molecule JIB-04 disrupts O(2) binding in the Fe-dependent histone demethylase KDM4A/JMJD2A()

JIB-04, a specific inhibitor of the O(2)-activating, Fe-dependent histone lysine demethylases, is revealed to disrupt the binding of O(2) in KDM4A/JMJD2A through a continuous O(2)-consumption assay, X-ray crystal structure data, and molecular docking.

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Detalhes bibliográficos
Publicado no:Chem Commun (Camb)
Main Authors: Cascella, Barbara, Lee, Soon Goo, Singh, Sukrit, Jez, Joseph M., Mirica, Liviu M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5511625/
https://ncbi.nlm.nih.gov/pubmed/28144654
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6cc09882g
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