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Chiral Brønsted Acid‐Catalyzed Asymmetric Synthesis of N‐Aryl‐cis‐aziridine Carboxylate Esters

We report a multi‐component asymmetric Brønsted acid‐catalyzed aza‐Darzens reaction which is not limited to specific aromatic or heterocyclic aldehydes. Incorporating alkyl diazoacetates and, important for high ee's, ortho‐tert‐butoxyaniline our optimized reaction (i.e. solvent, temperature and...

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Bibliografiske detaljer
Udgivet i:Angew Chem Int Ed Engl
Main Authors: Bew, Sean P., Liddle, John, Hughes, David L., Pesce, Paolo, Thurston, Sean M.
Format: Artigo
Sprog:Inglês
Udgivet: John Wiley and Sons Inc. 2017
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5502890/
https://ncbi.nlm.nih.gov/pubmed/28378388
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201611990
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