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Factors influencing biased agonism in recombinant cells expressing the human α(1A)‐adrenoceptor
BACKGROUND AND PURPOSE: Agonists acting at GPCRs promote biased signalling via Gα or Gβγ subunits, GPCR kinases and β‐arrestins. Since the demonstration of biased agonism has implications for drug discovery, it is essential to consider confounding factors contributing to bias. We have examined bias...
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| Publicado no: | Br J Pharmacol |
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| Main Authors: | , , , , , , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
John Wiley and Sons Inc.
2017
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5481649/ https://ncbi.nlm.nih.gov/pubmed/28444738 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.13837 |
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