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Parallelized Ligand Screening Using Dissolution Dynamic Nuclear Polarization

Protein−ligand interactions are frequently screened using nuclear magnetic resonance (NMR) spectroscopy. The dissociation constant (K(D)) of a ligand of interest can be determined via a spin-spin relaxation measurement of a reporter ligand, in a single scan when using hyperpolarization by means of d...

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Publicat a:Anal Chem
Autors principals: Kim, Yaewon, Liu, Mengxiao, Hilty, Christian
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5464406/
https://ncbi.nlm.nih.gov/pubmed/27723298
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.analchem.6b03382
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