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In Vitro Metabolism of Oprozomib, an Oral Proteasome Inhibitor: Role of Epoxide Hydrolases and Cytochrome P450s

Oprozomib is an oral proteasome inhibitor currently under investigation in patients with hematologic malignancies or solid tumors. Oprozomib elicits potent pharmacological actions by forming a covalent bond with the active site N-terminal threonine of the 20S proteasome. Oprozomib has a short half-l...

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Publicat a:Drug Metab Dispos
Autors principals: Wang, Zhican, Fang, Ying, Teague, Juli, Wong, Hansen, Morisseau, Christophe, Hammock, Bruce D., Rock, Dan A., Wang, Zhengping
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5452678/
https://ncbi.nlm.nih.gov/pubmed/28428366
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.117.075226
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