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Design and Synthesis of Potent and Selective PIM Kinase Inhibitors by Targeting Unique Structure of ATP-Binding Pocket

[Image: see text] In the development of kinase inhibitors, one of the major concerns is selectivity. An effective strategy to achieve high selectivity is to utilize structural differences among kinases to inform inhibitor design. Here, we set out to improve the PIM (proviral integration site for Mol...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Nakano, Hirofumi, Hasegawa, Tsukasa, Kojima, Hirotatsu, Okabe, Takayoshi, Nagano, Tetsuo
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2017
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5430388/
https://ncbi.nlm.nih.gov/pubmed/28523101
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.6b00518
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