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Synthesis and Evaluation of Novel Inhibitors of Pim-1 and Pim-2 Protein Kinases

The Pim protein kinases are frequently overexpressed in prostate cancer and certain forms of leukemia and lymphoma. 5-(3-Trifluoromethylbenzylidene)thiazolidine-2,4-dione (4a) was identified by screening to be a Pim-1 inhibitor and was found to attenuate the autophosphorylation of tagged Pim-1 in in...

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Publicado en:J Med Chem
Autores principales: Xia, Zuping, Knaak, Christian, Ma, Jian, Beharry, Zanna M., McInnes, Campbell, Wang, Wenxue, Kraft, Andrew S., Smith, Charles D.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2009
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5404933/
https://ncbi.nlm.nih.gov/pubmed/19072652
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm800937p
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