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Structural Features and Inhibitors of Bromodomains

Bromodomains are conserved structural modules responsible for recognizing acetylated-lysine residues on histone tails and other transcription-associated proteins, such as transcription factors and co-factors. Owing to their important functions in the regulation of ordered gene transcription in chrom...

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Dettagli Bibliografici
Pubblicato in:Drug Discov Today Technol
Autori principali: Meslamani, Jamel, Smith, Steven G., Sanchez, Roberto, Zhou, Ming-Ming
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5325140/
https://ncbi.nlm.nih.gov/pubmed/27769355
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ddtec.2016.09.001
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