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Dynamic Structure and Inhibition of a Malaria Drug Target: Geranylgeranyl Diphosphate Synthase

We report a molecular dynamics investigation of the structure, function and inhibition of geranylgeranyl diphosphate synthase (GGPPS), a potential drug target, from the malaria parasite Plasmodium vivax. We discovered several GGPPS inhibitors, benzoic acids, and solved their structures crystallograp...

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Dades bibliogràfiques
Publicat a:Biochemistry
Autors principals: Ricci, Clarisse G., Liu, Yi-Liang, Zhang, Yonghui, Wang, Yang, Zhu, Wei, Oldfield, Eric, McCammon, J. Andrew
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5319852/
https://ncbi.nlm.nih.gov/pubmed/27564465
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.6b00398
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