Загрузка...

Total synthesis of a key series of vinblastines modified at C4 that define the importance and surprising trends in activity

The total synthesis and evaluation of a key systematic series of vinblastines that incorporate the first deep-seated changes to the substituent at C4 are detailed. The synthetic approach features an expanded and redefined scope of a 1,3,4-oxadiazole [4 + 2]/[3 + 2] cycloaddition cascade in which ele...

Полное описание

Сохранить в:
Библиографические подробности
Опубликовано в: :Chem Sci
Главные авторы: Yang, Shouliang, Sankar, Kuppusamy, Skepper, Colin K., Barker, Timothy J., Lukesh III, John C., Brody, Daniel M., Brütsch, Manuela M., Boger, Dale L.
Формат: Artigo
Язык:Inglês
Опубликовано: Royal Society of Chemistry 2017
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5302862/
https://ncbi.nlm.nih.gov/pubmed/28194270
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c6sc04146a
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!