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Mocetinostat (MGCD0103): a review of an isotype-specific histone deacetylase inhibitor

INTRODUCTION: HDAC inhibitors (HDACIs) have the potential to restore gene expression and display antitumor effects in vitro. As single agents, HDACIs have clinical activity in lymphoma. In myeloid leukemias, combinations of DNA methylation inhibitors and HDACIs are promising. Other combinations are...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Expert Opin Investig Drugs
Egile Nagusiak: Boumber, Yanis, Younes, Anas, Garcia-Manero, Guillermo
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2011
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC5206967/
https://ncbi.nlm.nih.gov/pubmed/21554162
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/13543784.2011.577737
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