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Mocetinostat (MGCD0103): a review of an isotype-specific histone deacetylase inhibitor

INTRODUCTION: HDAC inhibitors (HDACIs) have the potential to restore gene expression and display antitumor effects in vitro. As single agents, HDACIs have clinical activity in lymphoma. In myeloid leukemias, combinations of DNA methylation inhibitors and HDACIs are promising. Other combinations are...

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Publicado en:Expert Opin Investig Drugs
Main Authors: Boumber, Yanis, Younes, Anas, Garcia-Manero, Guillermo
Formato: Artigo
Idioma:Inglês
Publicado: 2011
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5206967/
https://ncbi.nlm.nih.gov/pubmed/21554162
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/13543784.2011.577737
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