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Mocetinostat (MGCD0103): a review of an isotype-specific histone deacetylase inhibitor

INTRODUCTION: HDAC inhibitors (HDACIs) have the potential to restore gene expression and display antitumor effects in vitro. As single agents, HDACIs have clinical activity in lymphoma. In myeloid leukemias, combinations of DNA methylation inhibitors and HDACIs are promising. Other combinations are...

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Enregistré dans:
Détails bibliographiques
Publié dans:Expert Opin Investig Drugs
Auteurs principaux: Boumber, Yanis, Younes, Anas, Garcia-Manero, Guillermo
Format: Artigo
Langue:Inglês
Publié: 2011
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5206967/
https://ncbi.nlm.nih.gov/pubmed/21554162
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/13543784.2011.577737
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