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In vitro to in vivo extrapolation of the complex drug-drug interaction of bupropion and its metabolites with CYP2D6; simultaneous reversible inhibition and CYP2D6 downregulation

Bupropion is a widely used antidepressant and smoking cessation aid and a strong inhibitor of CYP2D6 in vivo. Bupropion is administered as a racemic mixture of R- and S-bupropion and has stereoselective pharmacokinetics. Four primary metabolites of bupropion, threo- and erythrohydrobupropion and R,R...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Biochem Pharmacol
Päätekijät: Sager, Jennifer E., Tripathy, Sasmita, Price, Lauren SL., Nath, Abhinav, Chang, Justine, Stephenson-Famy, Alyssa, Isoherranen, Nina
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2016
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC5164944/
https://ncbi.nlm.nih.gov/pubmed/27836670
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2016.11.007
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