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Tamoxifen Isomers and Metabolites Exhibit Distinct Affinity and Activity at Cannabinoid Receptors: Potential Scaffold for Drug Development

Tamoxifen (Tam) is a selective estrogen receptor (ER) modulator (SERM) that is an essential drug to treat ER-positive breast cancer. Aside from known actions at ERs, recent studies have suggested that some SERMs like Tam also exhibit novel activity at cannabinoid subtype 1 and 2 receptors (CB1R and...

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Publicat a:PLoS One
Autors principals: Ford, Benjamin M., Franks, Lirit N., Radominska-Pandya, Anna, Prather, Paul L.
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5147891/
https://ncbi.nlm.nih.gov/pubmed/27936172
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0167240
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