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Tramadol Metabolism to O-Desmethyl Tramadol (M1) and N-Desmethyl Tramadol (M2) by Dog Liver Microsomes: Species Comparison and Identification of Responsible Canine Cytochrome P450s

Tramadol is widely used to manage mild to moderately painful conditions in dogs. However, this use is controversial, since clinical efficacy studies in dogs showed conflicting results, whereas pharmacokinetic studies demonstrated relatively low circulating concentrations of O-desmethyltramadol (M1)....

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Foilsithe in:Drug Metab Dispos
Main Authors: Perez, Tania E., Mealey, Katrina L., Grubb, Tamara L., Greene, Stephen A., Court, Michael H.
Formáid: Artigo
Teanga:Inglês
Foilsithe: The American Society for Pharmacology and Experimental Therapeutics 2016
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Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5118633/
https://ncbi.nlm.nih.gov/pubmed/27758804
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.071902
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