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Tramadol Metabolism to O-Desmethyl Tramadol (M1) and N-Desmethyl Tramadol (M2) by Dog Liver Microsomes: Species Comparison and Identification of Responsible Canine Cytochrome P450s

Tramadol is widely used to manage mild to moderately painful conditions in dogs. However, this use is controversial, since clinical efficacy studies in dogs showed conflicting results, whereas pharmacokinetic studies demonstrated relatively low circulating concentrations of O-desmethyltramadol (M1)....

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Dades bibliogràfiques
Publicat a:Drug Metab Dispos
Autors principals: Perez, Tania E., Mealey, Katrina L., Grubb, Tamara L., Greene, Stephen A., Court, Michael H.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5118633/
https://ncbi.nlm.nih.gov/pubmed/27758804
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.071902
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