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Exploration of the conformational landscape in pregnane X receptor reveals a new binding pocket

Ligand‐regulated pregnane X receptor (PXR), a member of the nuclear receptor superfamily, plays a central role in xenobiotic metabolism. Despite its critical role in drug metabolism, PXR activation can lead to adverse drug‐drug interactions and early stage metabolism of drugs. Activated PXR can indu...

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Библиографические подробности
Опубликовано в: :Protein Sci
Главные авторы: Chandran, Aneesh, Vishveshwara, Saraswathi
Формат: Artigo
Язык:Inglês
Опубликовано: John Wiley and Sons Inc. 2016
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5079256/
https://ncbi.nlm.nih.gov/pubmed/27515410
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/pro.3012
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