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Design, Synthesis, and Antitumor Evaluation of 4-Amino-(1H)-pyrazole Derivatives as JAKs Inhibitors

[Image: see text] Abnormalities in the JAK/STAT signaling pathway lead to many diseases such as immunodeficiency, inflammation, and cancer. Herein, we designed and synthesized a series of 4-amino-(1H)-pyrazole derivatives as potent JAKs inhibitors for cancer treatment. Results from in vitro protein...

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Pubblicato in:ACS Med Chem Lett
Autori principali: Liang, Xuewu, Zang, Jie, Zhu, Mengyuan, Gao, Qianwen, Wang, Binghe, Xu, Wenfang, Zhang, Yingjie
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2016
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5066150/
https://ncbi.nlm.nih.gov/pubmed/27774135
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.6b00247
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