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Pharmacokinetic–pharmacodynamic modelling of drug‐induced QTc interval prolongation in man: prediction from in vitro human ether‐à‐go‐go‐related gene binding and functional inhibition assays and conscious dog studies

BACKGROUND AND PURPOSE: Functional measures of human ether‐à‐go‐go‐related gene (hERG; K(v)11.1) channel inhibition have been prioritized as an in vitro screening tool for candidate molecules. However, it is unclear how these results can be translated to humans. Here, we explore how data on drug bin...

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Detalhes bibliográficos
Publicado no:Br J Pharmacol
Main Authors: Dubois, V F S, Casarotto, E, Danhof, M, Della Pasqua, O
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5055135/
https://ncbi.nlm.nih.gov/pubmed/27427789
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.13558
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