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Nitrotriazole-based acetamides and propanamides with broad spectrum antitrypanosomal activity
3-Nitro-1H-1,2,4-triazole-based acetamides bearing a biphenyl- or a phenoxyphenyl moiety have shown remarkable antichagasic activity both in vitro and in an acute murine model, as well as substantial in vitro antileishmanial activity but lacked activity against human African trypanosomiasis. We have...
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| Publicado no: | Eur J Med Chem |
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| Main Authors: | , , , , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
Editions Scientifiques Elsevier
2016
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5049494/ https://ncbi.nlm.nih.gov/pubmed/27543881 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2016.08.002 |
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