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Comparison of [(11)C]TZ1964B and [(18)F]MNI659 for PET imaging brain PDE10A in nonhuman primates

Phosphodiesterase 10A (PDE10A) inhibitors show therapeutic effects for diseases with striatal pathology. PET radiotracers have been developed to quantify in vivo PDE10A levels and target engagement for therapeutic interventions. The aim of this study was to compare two potent and selective PDE10A ra...

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Dettagli Bibliografici
Pubblicato in:Pharmacol Res Perspect
Autori principali: Liu, Hui, Jin, Hongjun, Yue, Xuyi, Han, Junbin, Yang, Hao, Flores, Hubert, Su, Yi, Alagille, David, Perlmutter, Joel S., Tamagnan, Gilles, Tu, Zhude
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2016
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5045939/
https://ncbi.nlm.nih.gov/pubmed/27713824
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.253
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