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Histone deacetylase 6 structure and molecular basis of catalysis and inhibition

Histone deacetylase 6 (HDAC6) is a critical target for drug design due to its role in oncogenic transformation and cancer metastasis, and is unique among all histone deacetylases in that it contains tandem catalytic domains designated CD1 and CD2. We now report the crystal structures of CD2 from Hom...

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Detalhes bibliográficos
Publicado no:Nat Chem Biol
Main Authors: Hai, Yang, Christianson, David W.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4990478/
https://ncbi.nlm.nih.gov/pubmed/27454933
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.2134
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