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Molecular Basis for the Selective Inhibition of Histone Deacetylase 6 by a Mercaptoacetamide Inhibitor

[Image: see text] Mercaptoacetamide histone deacetylase inhibitors are neuroprotective agents that do not exhibit the genotoxicity associated with more commonly used hydroxamate inhibitors. Here, we present the crystal structure of a selective mercaptoacetamide complexed with the C-terminal catalyti...

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Библиографические подробности
Опубликовано в: :ACS Med Chem Lett
Главные авторы: Porter, Nicholas J., Shen, Sida, Barinka, Cyril, Kozikowski, Alan P., Christianson, David W.
Формат: Artigo
Язык:Inglês
Опубликовано: American Chemical Society 2018
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6295862/
https://ncbi.nlm.nih.gov/pubmed/30613344
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00487
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