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Discovery and characterization of novel small-molecule CXCR4 receptor agonists and antagonists

The chemokine CXCL12 (SDF-1) and its cognate receptor CXCR4 are involved in a large number of physiological processes including HIV-1 infectivity, inflammation, tumorigenesis, stem cell migration, and autoimmune diseases. While previous efforts have identified a number of CXCR4 antagonists, there ha...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Mishra, Rama K., Shum, Andrew K., Platanias, Leonidas C., Miller, Richard J., Schiltz, Gary E.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4960487/
https://ncbi.nlm.nih.gov/pubmed/27456816
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep30155
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