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Macrocyclic Envelope Glycoprotein Antagonists that Irreversibly Inactivate HIV-1 before Host Cell Encounter

We derived macrocyclic HIV-1 antagonists as a new class of peptidomimetic drug leads. Cyclic peptide triazoles (cPTs) retained the gp120 inhibitory and virus-inactivating signature of parent PTs, arguing that cyclization locked an active conformation. The 6-residue cPT 9 (AAR029b) exhibited sub-micr...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Rashad, Adel A., Sundaram, Ramalingam Venkat Kalyana, Aneja, Rachna, Duffy, Caitlin, Chaiken, Irwin
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4936186/
https://ncbi.nlm.nih.gov/pubmed/26331669
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b00935
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